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Medications used to treat lower urinary symptoms attributed to benign prostatic hyperplasia
Drug class Medication
Alpha-1 blockers (ABs)
  • Silodosin (Rapaflo)
  • Terazosin (Hytrin)
  • Alfuzosin (Uroxatral)
  • Doxazosin (Cardura)
  • Tamsulosin (Flomax)
5-alpha-reductase inhibitors (5-ARIs)
  • Finasteride (Proscar)
  • Dutasteride (Avodart)
Anticholinergic agents
  • Oxybutynin (Oxytrol)
  • Fesoterodine (Toviaz)
  • Darifenacin (Enablex)
  • Tolterodine (Detrol, Detrol LA)
  • Solifenacin (VESIcare)
  • Trospium (Sanctura)
Beta-3 adrenergic agonist
  • Mirabegron (Myrbetriq)
Phosphodiesterase type 5 (PDE-5) inhibitors
  • Tadalafil (Cialis)
  • Sildenafil (Viagra)
  • Avanafil (Stendra)
  • Vardenafil (Staxyn, Levitra)
Adapted from: Brasure M, MacDonald R, Dahm P, et al. Newer medications for lower urinary tract symptoms attributed to benign prostatic hyperplasia: A review. Comparative Effectiveness Review No. 178, AHRQ Publication No. 16-EHC024-EF, Agency for Healthcare Research and Quality, Rockville, MD 2016.
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